Time slot | Speaker | Topic | Location |
08.00-09.00 | Gerhard Mueller | Medicinal Chemistry Targeted Towards the Kinase Family | auditorium |
09.00-10.00 | Andrew Mortlock | Targeting the hallmarks of cancer – medicinal chemistry beyond the kinome | auditorium |
10.00-10.30 | Coffee break | ||
10.30-11.30 | Tjeerd Barf | Irreversible Kinase Inhibitor Drugs | auditorium |
11.30-13.00 | Lunch |
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13.00-15.15 | S. Gremmen/ J. Slootweg/ M. Carneiro |
T1: Hit Finding in Today’s Target Space | |
M. Eerland/ C. Commandeur |
T1: From Hit to New Drug | ||
13.00-15.15 | A. Mortlock | T2: Developing a Lead | |
N. Meanwell/ M. Commandeur |
T2: Applications of Bioisosteres in Drug Design | ||
13.00-15.15 | M. Whittaker/ M. Mazanetz |
T3: Fragment Based Drug Discovery | |
J. Viklund/ F. Karlsson |
T3: Structure-Based Drug Design | ||
15.30-23.30 | Special event: Guided tour and wine tasting in Aigle Castle, course dinner |