Time slot	Speaker	Topic	Location
08.00-09.00	Karin Briner	To be announced	auditorium
09.00-10.00	Adrian Whitty	Macrocycles and Other Beyond Rule-of-5 Chemotypes: Opportunities and Challenges	auditorium
10.00-10.30	Coffee break
10.30-11.30	Andrea Decker	“Drug-Likeness”: Physicochemical Properties in Small-Molecule Drug Discovery	auditorium
11.30-12.30	Brian Shoichet	Colloidal Aggregation and Chemical Space in Early Discovery	auditorium
12.30-13.30	Lunch
14.00-15.00	Karl-Heinz Altmann	Natural Product – Based Drug Discovery	auditorium
15.30-17.45	S. Gremmen/ J. Slootweg/ M. Carneiro	T1: Hit Finding in Today’s Target Space
	M. Eerland/ C. Commandeur	T1: From Hit to New Drug
15.30-17.45	A. Mortlock	T2: Developing a Lead
	N. Meanwell/ M. Commandeur	T2: Applications of Bioisosteres in Drug Design
15.30-17.45	M. Whittaker/ M. Mazanetz	T3: Fragment Based Drug Discovery
	J. Viklund/ F. Karlsson	T3: Structure-Based Drug Design
18.00-19.00	Gerhard Klebe	What Thermodynamics Can Help to Understand Protein-Ligand Binding in Medicinal Chemistry	auditorium
19.00-20.30	Dinner
20.30-21.30	Jason McCartney	Discovery of CFTR Modulators for Cystic Fibrosis	auditorium